SCHEMBL21295033

SCHEMBL21295033

CC(C)(C)NC(=O)OC1CNc2ccccc2C1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.56
MTNR1A P48039 1/20 0.49
MTNR1B P49286 1/20 0.49
MAPK1 P28482 6/20 0.39
SIRT2 Q8IXJ6 1/20 0.39
CCNE1 P24864 2/20 0.37
CDK2 P24941 2/20 0.37
GSK3B P49841 1/20 0.37
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
TACR1 P25103 1/20 0.35
ANO1 Q5XXA6 1/20 0.35
BRD4 O60885 1/20 0.34
DPP8 Q6V1X1 1/20 0.34
DPP9 Q86TI2 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8564559 0.85 EPHX2 (0.53) EPHX2MTNR1AMTNR1BMAPK1GAA
SCHEMBL8564566 0.85 EPHX2 (0.53) EPHX2MTNR1AMTNR1BMAPK1GAA
SCHEMBL8564568 0.85 EPHX2 (0.53) EPHX2MTNR1AMTNR1BMAPK1GAA
SCHEMBL17049225 0.83 EPHX2 (0.54) EPHX2MTNR1AMTNR1BMAPK1GAA
SCHEMBL28791460 0.83 FABP7 (0.43) EPHX2MTNR1AMTNR1BTACR1ANO1
SCHEMBL8562145 0.80 MTNR1A (0.56) EPHX2MTNR1AMTNR1BMAPK1GAA
SCHEMBL8562147 0.80 MTNR1A (0.56) EPHX2MTNR1AMTNR1BMAPK1GAA
SCHEMBL8562150 0.80 MTNR1A (0.56) EPHX2MTNR1AMTNR1BMAPK1GAA
SCHEMBL8086570 0.79 MTNR1A (0.50) EPHX2MTNR1AMTNR1BMAPK1GAA
SCHEMBL9036114 0.79 MTNR1A (0.50) EPHX2MTNR1AMTNR1BMAPK1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116783165-A 1,2,3, 4-tetrahydroquinoline derivatives as YAP/TAZ-TEAD activation inhibitors for the treatment of cancer 天主教鲁汶大学 2023-09-19 CN disclosed
WO-2019161803-A1 PEPTIDYLARGININE DEIMINASE INHIBITOR AND USE THEREOF 南京药捷安康生物科技有限公司 2019-08-29 WO disclosed