SCHEMBL21296484

SCHEMBL21296484

O=C[C@@H](Br)Cc1ccccc1Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.42
PNMT P11086 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
PPARG P37231 1/20 0.40
PPARA Q07869 1/20 0.40
TAAR1 Q96RJ0 3/20 0.39
RAB9A P51151 2/20 0.39
NPC1 O15118 1/20 0.39
CHRM2 P08172 1/20 0.39
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
SLC6A3 Q01959 2/20 0.38
LMNA P02545 2/20 0.37
DAO P14920 1/20 0.37
PKM P14618 1/20 0.36
HTT P42858 1/20 0.36
MEN1 O00255 1/20 0.36
TP53 P04637 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL232677 0.78 IDO1 (0.43) IDO1PNMTSMN1; SMN2PPARGPPARA
SCHEMBL1922202 0.78 IDO1 (0.46) IDO1SMN1; SMN2RAB9ANPC1SLC6A4
SCHEMBL9480317 0.77 IDO1 (0.50) IDO1PNMTSMN1; SMN2PPARGPPARA
SCHEMBL30461921 0.77 SLC6A2 (0.50) IDO1PNMTSMN1; SMN2PPARGPPARA
SCHEMBL16298056 0.77 SLC6A2 (0.50) IDO1PNMTSMN1; SMN2PPARGPPARA
SCHEMBL14237917 0.77 SLC6A2 (0.50) IDO1PNMTSMN1; SMN2PPARGPPARA
SCHEMBL16463838 0.77 SLC6A2 (0.46) IDO1PNMTSMN1; SMN2PPARGPPARA
SCHEMBL4764946 0.77 ALDH1A1 (0.41) IDO1SMN1; SMN2PPARGPPARATAAR1
SCHEMBL14208189 0.77 SLC6A2 (0.46) IDO1PNMTSMN1; SMN2PPARGPPARA
SCHEMBL5238119 0.76 MEN1 (0.32) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3755699-A1 SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF Relay Therapeutics, Inc. (US) 2020-12-30 EP disclosed
WO-2019165073-A1 SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. (US) 2019-08-29 WO disclosed