SCHEMBL4764946

SCHEMBL4764946

O=CC(Br)Cc1ccccc1F

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
TAAR1 Q96RJ0 3/20 0.41
LMNA P02545 1/20 0.39
IDO1 P14902 2/20 0.38
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
KCNH2 Q12809 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
DAO P14920 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21296484 0.77 IDO1 (0.42) TAAR1LMNAIDO1PPARGPPARA
SCHEMBL21395226 0.77 PPARG (0.41) ALDH1A1TAAR1LMNAIDO1PPARG
SCHEMBL14640229 0.77 TAAR1 (0.45) ALDH1A1TAAR1LMNAIDO1PPARG
SCHEMBL14640355 0.77 ALDH1A1 (0.41) ALDH1A1TAAR1LMNAIDO1PPARG
SCHEMBL8433364 0.77 TAAR1 (0.45) ALDH1A1TAAR1LMNAIDO1PPARG
SCHEMBL6153079 0.77 ALDH1A1 (0.41) ALDH1A1TAAR1LMNAIDO1PPARG
SCHEMBL6200983 0.75 TAAR1 (0.46) ALDH1A1TAAR1LMNAIDO1PPARG
SCHEMBL5211715 0.75 TAAR1 (0.46) ALDH1A1TAAR1LMNAIDO1PPARG
SCHEMBL4269883 0.75 NAPRT (0.36)
SCHEMBL19812660 0.74 TAAR1 (0.47) ALDH1A1TAAR1LMNAIDO1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919865-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2008-05-14 EP disclosed
WO-2007026916-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-08 WO disclosed