SCHEMBL21301600

SCHEMBL21301600

COC(=O)C(CC(C)C)NCc1ccc(N)cc1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PPID Q08752 2/20 0.57
ITGB1 P05556 3/20 0.49
ITGA5 P08648 3/20 0.49
TAS1R3 Q7RTX0 9/20 0.48
TAS1R1 Q7RTX1 9/20 0.48
ITGB3 P05106 2/20 0.47
ITGAV P06756 2/20 0.47
CTSK P43235 1/20 0.46
ANPEP P15144 2/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
PPIB P23284 1/20 0.42
PPIA P62937 1/20 0.42
PPIG Q13427 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3957241 0.85 NOS3 (0.55) PPIDTAS1R3TAS1R1CTSKANPEP
SCHEMBL24446769 0.85 ANPEP (0.59) TAS1R3TAS1R1CTSKANPEP
SCHEMBL3955671 0.85 NOS3 (0.55) PPIDTAS1R3TAS1R1CTSKANPEP
SCHEMBL3955674 0.85 NOS3 (0.55) PPIDTAS1R3TAS1R1CTSKANPEP
SCHEMBL20447100 0.85 ANPEP (0.59) TAS1R3TAS1R1CTSKANPEP
SCHEMBL19975277 0.85 ATM (0.54) TAS1R3TAS1R1CTSKANPEPCA12
SCHEMBL7365655 0.85 ATM (0.54) TAS1R3TAS1R1CTSKANPEPCA12
SCHEMBL6129757 0.85 ATM (0.54) TAS1R3TAS1R1CTSKANPEPCA12
SCHEMBL27723661 0.85 ITGB1 (0.55) PPIDITGB1ITGA5ITGB3ITGAV
SCHEMBL27723663 0.85 ITGB1 (0.55) PPIDITGB1ITGA5ITGB3ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3530290-A1 ALPHA AMINOACID ESTER-DRUG CONJUGATES HYDROLYSABLE BY CARBOXYLESTERASE GlaxoSmithKline Intellectual Property Development Limited (GB) 2019-08-28 EP disclosed