SCHEMBL21303003

SCHEMBL21303003

COc1nc(Cl)nc2c1cnn2COCC[Si](C)(C)C

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.32
DGAT1 O75907 1/20 0.32
PNP P00491 2/20 0.32
HSP90AA1 P07900 1/20 0.31
TRAP1 Q12931 1/20 0.31
CNR2 P34972 1/20 0.30
PDE2A O00408 1/20 0.30
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29661419 0.87 HSP90AA1 (0.35) MAPTDGAT1PNPHSP90AA1TRAP1
SCHEMBL24328469 0.87 HSP90AA1 (0.35) MAPTDGAT1PNPHSP90AA1TRAP1
SCHEMBL25875898 0.85 MAPT (0.33) MAPTDGAT1PNPPDE2A
SCHEMBL21481639 0.84 NT5E (0.38) MAPTDGAT1PNPHSP90AA1TRAP1
SCHEMBL30982195 0.78 DGAT1 (0.33) MAPTDGAT1HSP90AA1CYP1A2
SCHEMBL26720567 0.77 HSP90AA1 (0.36) MAPTDGAT1PNPHSP90AA1TRAP1
SCHEMBL20262422 0.76 DGAT1 (0.33) MAPTDGAT1
SCHEMBL26102605 0.74 BCDIN3D (0.42) MAPTPDE2ACYP1A2
SCHEMBL21398946 0.74
SCHEMBL4015126 0.74 ABL1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200392161-A1 SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF SCHRÖDINGER, INC. 2020-12-17 US disclosed
US-20200392161-A1 SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF SCHRÖDINGER, INC. 2020-12-17 US disclosed
WO-2019165073-A1 SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. (US) 2019-08-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200392161-A1 SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF PTPRCAP, PTPRJ, PTPRC MAPT 4383/4885DGAT1 890/4885PNP 1400/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.