SCHEMBL21481639

SCHEMBL21481639

C[Si](C)(C)CCOCn1ncc2c(N)nc(Cl)nc21

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NT5E P21589 2/20 0.38
PNP P00491 2/20 0.36
CYP3A4 P08684 6/20 0.36
CYP2D6 P10635 4/20 0.35
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
MAPT P10636 1/20 0.32
CDK1 P06493 1/20 0.32
HSP90AA1 P07900 1/20 0.31
TRAP1 Q12931 1/20 0.31
PDE2A O00408 1/20 0.31
NPC1 O15118 1/20 0.31
DGAT1 O75907 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24328469 0.88 HSP90AA1 (0.35) PNPADORA3ADORA2AADORA1MAPT
SCHEMBL29661419 0.88 HSP90AA1 (0.35) PNPADORA3ADORA2AADORA1MAPT
SCHEMBL30041757 0.87 PNP (0.38) PNPCYP3A4CYP2D6ADORA2AADORA1
SCHEMBL25875898 0.86 MAPT (0.33) PNPMAPTPDE2ADGAT1
SCHEMBL21303003 0.84 MAPT (0.32) PNPMAPTHSP90AA1TRAP1PDE2A
SCHEMBL26720567 0.78 HSP90AA1 (0.36) PNPMAPTHSP90AA1TRAP1NPC1
SCHEMBL20262422 0.77 DGAT1 (0.33) MAPTDGAT1
SCHEMBL21462203 0.77 NPC1 (0.37) NT5EMAPTCDK1NPC1
SCHEMBL13737735 0.77 DGAT1 (0.34) NT5EMAPTCDK1HSP90AA1NPC1
SCHEMBL21462293 0.76 CYP3A4 (0.39) PNPCYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019196918-A1 FIVE-MEMBERED HETEROCYCLO-PYRIMIDINE COMPOUND, PHARMACEUTICAL COMPOSITION AND USE THEREOF 罗欣药业(上海)有限公司 2019-10-17 WO disclosed