SCHEMBL21311802

SCHEMBL21311802

Cn1c2c(c(=O)c3ccccc31)CCCC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.53
HTR2C P28335 1/20 0.53
KDM4E B2RXH2 5/20 0.51
HSD17B10 Q99714 3/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
ALOX15 P16050 1/20 0.51
MAPK1 P28482 1/20 0.51
HPGD P15428 4/20 0.51
LMNA P02545 1/20 0.51
ALOX5 P09917 1/20 0.50
PTGS1 P23219 1/20 0.50
PTGS2 P35354 1/20 0.50
ALDH1A1 P00352 4/20 0.47
HTT P42858 2/20 0.47
GLA P06280 1/20 0.47
GAA P10253 1/20 0.47
CYP2C19 P33261 1/20 0.47
NQO2 P16083 1/20 0.46
TSHR P16473 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3927394 0.87 HTR2A (0.67) HTR2AHTR2CKDM4EHSD17B10CYP1A2
SCHEMBL30223611 0.87 HTR2A (0.67) HTR2AHTR2CKDM4EHSD17B10CYP1A2
SCHEMBL15307679 0.86 HTR2A (0.65) HTR2AHTR2CKDM4EHSD17B10CYP1A2
SCHEMBL844491 0.84 HTR2A (0.67) HTR2AHTR2CKDM4EHSD17B10CYP1A2
SCHEMBL22879589 0.79 CA1 (0.45) KDM4EHSD17B10HPGDLMNAALDH1A1
SCHEMBL24119475 0.79 CA1 (0.42) HTR2AHTR2CKDM4EHSD17B10HPGD
SCHEMBL10309072 0.78 KDM4E (0.64) HTR2AHTR2CKDM4EHSD17B10CYP1A2
SCHEMBL7428637 0.78 HTR2A (0.51) HTR2AHTR2CKDM4EHSD17B10CYP1A2
SCHEMBL11463080 0.77 HTR2A (0.46) HTR2AHTR2CKDM4EHSD17B10CYP1A2
SCHEMBL11454621 0.77 HTR2A (0.50) HTR2AHTR2CKDM4EHSD17B10CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019161781-A1 RECEPTOR ANTAGONIST, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND USAGE THEREOF 北京泰德制药股份有限公司 2019-08-29 WO disclosed