SCHEMBL21336710

SCHEMBL21336710

COc1c(C)cnc2c(-c3ccc(C#N)cc3)cccc12

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.40
HPGDS O60760 1/20 0.39
CYP11B2 P19099 3/20 0.39
FYN P06241 1/20 0.38
IRAK4 Q9NWZ3 1/20 0.37
KDM4A O75164 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
KIT P10721 1/20 0.36
SCN8A Q9UQD0 1/20 0.36
CYP11B1 P15538 1/20 0.36
STAT3 P40763 1/20 0.36
PRKDC P78527 1/20 0.35
SLC22A12 Q96S37 1/20 0.35
PARP1 P09874 1/20 0.35
CTSA P10619 1/20 0.35
MAPKAPK2 P49137 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21336706 0.88 ALDH1A1 (0.39) HRH4HPGDSCYP11B2FYNIRAK4
SCHEMBL17128140 0.86 HRH4 (0.44) HRH4HPGDSCYP11B2FYNIRAK4
SCHEMBL17127609 0.86 HRH4 (0.39) HRH4HPGDSCYP11B2FYNIRAK4
SCHEMBL17127906 0.86 HRH4 (0.39) HRH4HPGDSCYP11B2FYNIRAK4
SCHEMBL17127785 0.84 SQOR (0.41) HRH4HPGDSCYP11B2FYNIRAK4
SCHEMBL17128379 0.84 HRH4 (0.38) HRH4HPGDSCYP11B2FYNIRAK4
SCHEMBL17128318 0.82 BRS3 (0.43) HRH4IRAK4KDM4AKDM5BSLC22A12
SCHEMBL17128200 0.81 HRH4 (0.41) HRH4HPGDSFYNIRAK4KDM4A
SCHEMBL17128203 0.81 IRAK4 (0.38) HRH4HPGDSFYNIRAK4KDM4A
SCHEMBL19001218 0.80 MEN1 (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3124482-B1 QUINOLINE DERIVATIVES AS SMO INHIBITORS GUANGDONG ZHONGSHENG PHARMACEUTICAL CO LTD (CN) 2019-09-11 EP disclosed