SCHEMBL21337541

SCHEMBL21337541

C=C(CC)N(CC1(N2CCN(CCc3cccnc3)CC2)CCOCC1)c1ccccn1

nearest known ligand 0.53

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 20/20 0.53
SIGMAR1 Q99720 19/20 0.53
KCNH2 Q12809 7/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19631785 0.78 OPRM1 (0.44) OPRM1SIGMAR1KCNH2
SCHEMBL18426780 0.77 SIGMAR1 (0.87) OPRM1SIGMAR1KCNH2
SCHEMBL18458749 0.77 OPRM1 (0.84) OPRM1SIGMAR1KCNH2
SCHEMBL21337545 0.74 SIGMAR1 (0.81) OPRM1SIGMAR1KCNH2
SCHEMBL18426573 0.74 OPRM1 (0.64) OPRM1SIGMAR1KCNH2
SCHEMBL18458333 0.74 SIGMAR1 (0.82) OPRM1SIGMAR1KCNH2
SCHEMBL20599205 0.73 OPRM1 (0.75) OPRM1SIGMAR1KCNH2
SCHEMBL18425865 0.73 SIGMAR1 (0.68) OPRM1SIGMAR1KCNH2
SCHEMBL19631711 0.73 OPRM1 (0.46) OPRM1SIGMAR1
SCHEMBL21337558 0.73 SIGMAR1 (0.73) OPRM1SIGMAR1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3328853-B1 SUBSTITUTED AMIDE DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN ESTEVE PHARMACEUTICALS SA (ES) 2019-09-11 EP disclosed