SCHEMBL21341963

SCHEMBL21341963

CCOC(=O)C1=C(c2ccc(OC)cc2)CN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.48
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
HPGD P15428 1/20 0.47
MAPT P10636 2/20 0.46
GPR119 Q8TDV5 1/20 0.44
CHRM5 P08912 3/20 0.42
CHRM1 P11229 3/20 0.42
P2RX3 P56373 1/20 0.42
HRH2 P25021 1/20 0.42
HRH1 P35367 1/20 0.42
SLC6A3 Q01959 1/20 0.42
HTT P42858 1/20 0.42
MMP1 P03956 3/20 0.41
MMP3 P08254 3/20 0.41
MMP7 P09237 3/20 0.41
MMP9 P14780 3/20 0.41
MMP8 P22894 3/20 0.41
MMP13 P45452 3/20 0.41
MMP2 P08253 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20476229 0.93 ALDH1A1 (0.50) ADORA1KDM4EALDH1A1HPGDGPR119
SCHEMBL14920560 0.92 CHRM5 (0.49) ADORA1KDM4EALDH1A1HPGDMAPT
SCHEMBL23040394 0.90 ALDH1A1 (0.47) ADORA1KDM4EALDH1A1HPGDGPR119
SCHEMBL14920221 0.88 ADORA1 (0.47) ADORA1MAPTCHRM5CHRM1HTT
SCHEMBL26647798 0.88 ALDH1A1 (0.47) ADORA1ALDH1A1MAPTCHRM5CHRM1
SCHEMBL26128665 0.88 ADORA1 (0.47) ADORA1KDM4EMAPTGPR119CHRM5
SCHEMBL23039761 0.88 ALDH1A1 (0.46) ADORA1KDM4EALDH1A1HPGDMAPT
SCHEMBL23632126 0.85 GPR119 (0.46) ADORA1GPR119CHRM5CHRM1HRH2
SCHEMBL23062407 0.85 GPR119 (0.47) ADORA1KDM4EALDH1A1HPGDMAPT
SCHEMBL23062601 0.85 MAPT (0.45) ADORA1KDM4EALDH1A1HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019170904-A1 PIPERIDINES OR PIPERIDONES SUBSTITUTED WITH UREA AND PHENYL Grünenthal GmbH (DE) 2019-09-12 WO disclosed