SCHEMBL21342033

SCHEMBL21342033

COc1cc(F)c([C@@H]2CN(C(=O)OC(C)(C)C)CCC2C(=O)O)c(F)c1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 3/20 0.45
ALDH1A1 P00352 1/20 0.44
GPR119 Q8TDV5 3/20 0.42
STS P08842 2/20 0.41
FPR1 P21462 3/20 0.41
DPP4 P27487 1/20 0.41
EPHX2 P34913 1/20 0.41
HTT P42858 1/20 0.40
USP30 Q70CQ3 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
FPR2 P25090 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21342468 1.00 PDE4B (0.45) PDE4BALDH1A1GPR119STSFPR1
SCHEMBL21342556 0.94 PDE4B (0.42) PDE4BALDH1A1GPR119STSDPP4
SCHEMBL21342312 0.87 ALDH1A1 (0.47) PDE4BALDH1A1GPR119STSEPHX2
SCHEMBL21342424 0.87 ALDH1A1 (0.47) PDE4BALDH1A1GPR119STSEPHX2
SCHEMBL21335089 0.87 DPP4 (0.42) PDE4BALDH1A1GPR119FPR1DPP4
SCHEMBL21341946 0.87 DPP4 (0.42) PDE4BALDH1A1GPR119FPR1DPP4
SCHEMBL23062474 0.85 PDE4B (0.42) PDE4BALDH1A1GPR119DPP4HTT
SCHEMBL21342337 0.84 YAP1 (0.43) PDE4BGPR119STSHTTUSP30
SCHEMBL23062607 0.81 ALDH1A1 (0.55) PDE4BALDH1A1GPR119STSHTT
SCHEMBL23062606 0.81 ALDH1A1 (0.55) PDE4BALDH1A1GPR119STSHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019170904-A1 PIPERIDINES OR PIPERIDONES SUBSTITUTED WITH UREA AND PHENYL Grünenthal GmbH (DE) 2019-09-12 WO disclosed