SCHEMBL21346321

SCHEMBL21346321

Cc1ccc(Cl)cc1CNC(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.41
SLC6A4 P31645 5/20 0.41
HTR2A P28223 4/20 0.41
OPRL1 P41146 1/20 0.40
CYP3A4 P08684 2/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39
POLB P06746 1/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 2/20 0.38
HSD17B10 Q99714 1/20 0.38
HIF1A Q16665 1/20 0.38
P2RX7 Q99572 1/20 0.36
TRPV4 Q9HBA0 1/20 0.36
ADRA2C P18825 1/20 0.36
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14438275 0.83 MEN1 (0.43) KCNH2SLC6A4HTR2AOPRL1CYP3A4
SCHEMBL2647752 0.79 MEN1 (0.57) KCNH2OPRL1CYP3A4MEN1CYP1A2
SCHEMBL25453552 0.79 MEN1 (0.43) SLC6A4CYP3A4MEN1CYP1A2CYP2D6
SCHEMBL12964268 0.79 SLC6A4 (0.59) KCNH2SLC6A4HTR2ASLC6A2SLC6A3
SCHEMBL21345583 0.77 LMNA (0.47) KCNH2SLC6A4HTR2AMEN1CYP1A2
SCHEMBL19862553 0.76 CXCR3 (0.43) KCNH2SLC6A4HTR2AOPRL1CYP3A4
SCHEMBL17449705 0.75 CYP3A4 (0.43) KCNH2SLC6A4HTR2ACYP3A4MEN1
SCHEMBL15432470 0.74 MEN1 (0.49) KCNH2SLC6A4HTR2ACYP3A4MEN1
SCHEMBL30995430 0.74 CYP3A4 (0.46) KCNH2SLC6A4HTR2ACYP3A4MEN1
SCHEMBL698696 0.74 CYP3A4 (0.46) KCNH2SLC6A4HTR2ACYP3A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019170086-A1 ACYL-SUBSTITUTED OXAZINO-QUINAZOLINE COMPOUND, PREPARATION METHOD THEREFOR, AND USES THEREOF 北京赛特明强医药科技有限公司 2019-09-12 WO disclosed