SCHEMBL21350985

SCHEMBL21350985

Cc1cc(Cl)ccc1-c1cc(C(=O)C(F)(F)F)sc1-c1ccc(Cl)cc1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 9/20 0.41
HDAC4 P56524 4/20 0.41
HDAC1 Q13547 6/20 0.37
GPBAR1 Q8TDU6 1/20 0.37
CYP2C9 P11712 1/20 0.37
HDAC3 O15379 2/20 0.37
RORC P51449 1/20 0.36
GRM2 Q14416 1/20 0.36
LMNA P02545 3/20 0.34
HTT P42858 3/20 0.34
MAPT P10636 2/20 0.34
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
HSP90AA1 P07900 1/20 0.34
KMT2A Q03164 1/20 0.34
TMPRSS4 Q9NRS4 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
TP53 P04637 1/20 0.34
ESR1 P03372 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26118486 0.87 HDAC6 (0.40) HDAC6HDAC4HDAC1GPBAR1CYP2C9
SCHEMBL12496481 0.83 DAO (0.47) GRM2MAPTMEN1KMT2AALDH1A1
SCHEMBL22901445 0.82 KDM4E (0.48) GRM2MAPTALDH1A1GAAESR1
SCHEMBL21350980 0.77 KDM4E (0.47) HDAC6HDAC4HDAC1HDAC3LMNA
SCHEMBL22901447 0.74 ESR2 (0.34) GPBAR1RORCGRM2LMNAHTT
SCHEMBL21350988 0.73 ESR2 (0.33) GPBAR1RORCGRM2ESR1ESR2
SCHEMBL21350986 0.70 GRM2 (0.36) GRM2LMNAMAPTKMT2AALDH1A1
SCHEMBL14310501 0.70 FLT1 (0.46) LMNAHTTMAPTMEN1POLB
SCHEMBL12497054 0.69 NOTUM (0.49) MAPTMEN1KMT2AALDH1A1TP53
SCHEMBL12496564 0.68 DAO (0.44) LMNAMAPTMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3762376-B1 DIPHENYL SUBSTITUTED THIOPHENE-2-AMIDE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS THEREOF USEFUL AS ANTIMICROBIAL DENOVAMED INC (CA) 2023-03-01 EP disclosed
WO-2019169479-A1 DIPHENYL SUBSTITUTED THIOPHENE-2-AMIDE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS THEREOF USEFUL AS ANTIMICROBIAL DENOVAMED INC. (CA) 2019-09-12 WO disclosed