SCHEMBL213577

SCHEMBL213577

O=CNc1cc(O)c2ccccc2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MYC P01106 1/20 0.41
MAX P61244 1/20 0.41
ERN1 O75460 2/20 0.41
LRRK2 Q5S007 2/20 0.39
MEN1 O00255 6/20 0.38
KMT2A Q03164 6/20 0.38
KDM4E B2RXH2 5/20 0.38
GAA P10253 4/20 0.38
MAPT P10636 4/20 0.38
POLB P06746 4/20 0.38
GFER P55789 4/20 0.38
L3MBTL1 Q9Y468 3/20 0.38
TDP1 Q9NUW8 2/20 0.38
HTT P42858 1/20 0.38
ALDH1A1 P00352 3/20 0.38
LMNA P02545 3/20 0.38
MAPK1 P28482 3/20 0.38
MMP14 P50281 2/20 0.38
THRB P10828 1/20 0.38
RECQL P46063 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28100413 0.81 SLC2A1 (0.46) ERN1MEN1KMT2AKDM4EMAPT
SCHEMBL27978560 0.80 LMNA (0.41) ERN1KMT2AKDM4EGAAMAPT
SCHEMBL27599847 0.79 PARP1 (0.40) MEN1KMT2AKDM4EGAAMAPT
SCHEMBL9071311 0.74 ERN1 (0.47) MYCMAXERN1MEN1KMT2A
SCHEMBL29951387 0.74 ERN1 (0.47) MYCMAXERN1MEN1KMT2A
SCHEMBL9731516 0.72 EGFR (0.44) MYCMAXERN1MEN1KMT2A
SCHEMBL9731511 0.72 MYC (0.37) MYCMAXERN1MEN1KMT2A
SCHEMBL557654 0.71 KDM1A (0.53) MEN1KMT2AKDM4EGAAMAPT
SCHEMBL29376440 0.70 MYC (0.52) MYCMAXMEN1KMT2AKDM4E
SCHEMBL9326676 0.70 MYC (0.52) MYCMAXMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106008373-B Disubstituted bicyclic derivative and its application as efflux pump inhibitor in antibacterial 山东大学 2019-02-22 CN disclosed
US-8088793-B2 Certain chemical entities, compositions, and methods CYTOKINETICS, INC. (US) 2012-01-03 US disclosed