SCHEMBL21360103

SCHEMBL21360103

Nc1cccc(C2C=CCC=C2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.42
CASP1 P29466 1/20 0.42
RECQL P46063 1/20 0.42
DDB1 Q16531 1/20 0.39
CRBN Q96SW2 1/20 0.39
ALDH1A1 P00352 4/20 0.36
CA1 P00915 3/20 0.35
CA2 P00918 3/20 0.35
CA9 Q16790 3/20 0.35
CA14 Q9ULX7 3/20 0.35
CA12 O43570 1/20 0.35
CA7 P43166 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
MAPT P10636 1/20 0.35
PTPN1 P18031 1/20 0.35
MAOA P21397 3/20 0.34
LMNA P02545 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21358187 0.76 CA12 (0.42) CYP3A4ALDH1A1CA2CA9CA14
SCHEMBL21358312 0.76 HTR2A (0.42) MAOAMAOBCYP19A1
SCHEMBL3740188 0.73 RECQL (0.39) CYP3A4RECQLMAOALMNATSHR
SCHEMBL21359879 0.73 HTR2C (0.51) CYP3A4DDB1CRBNALDH1A1CA1
SCHEMBL21358194 0.72 DRD2 (0.47) CASP1MAOATSHRENPP2MAOB
SCHEMBL29411064 0.70 CYP3A4 (0.50) CYP3A4CASP1RECQLDDB1CRBN
SCHEMBL273350 0.70 CYP3A4 (0.50) CYP3A4CASP1RECQLDDB1CRBN
SCHEMBL27660071 0.69 CYP3A4 (0.44) CYP3A4CASP1RECQLDDB1CRBN
Hydrochloric Acid SCHEMBL25305777 0.68 CYP3A4 (0.48) CYP3A4CASP1RECQLDDB1CRBN
SCHEMBL21250295 0.68 CYP3A4 (0.48) CYP3A4CASP1RECQLDDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019177117-A1 DRUG FOR TREATING COUGH 日本ケミファ株式会社 2019-09-19 WO claimed
WO-2019177117-A1 DRUG FOR TREATING COUGH 日本ケミファ株式会社 2019-09-19 WO disclosed
CN-103237794-A P2X4Receptor antagonists NIPPONCHEMIPHAR CO LTD 2013-08-07 CN disclosed