SCHEMBL21361262

SCHEMBL21361262

COc1cc(-c2ccc(F)cc2)cc(C)c1C1C(=O)CC2(CCN(C(=O)NC(=O)c3ccccn3)CC2)CC1O

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 13/20 0.36
KCNH2 Q12809 2/20 0.36
CCR8 P51685 1/20 0.36
GRIN2B Q13224 1/20 0.35
GRM4 Q14833 2/20 0.35
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
TLR7 Q9NYK1 1/20 0.33
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22859737 0.89 KCNH2 (0.38) CD274KCNH2CCR8GRIN2BGRM4
SCHEMBL21361250 0.84 MAOB (0.38) GRM4TLR7NPC1
SCHEMBL24120312 0.83 KCNH2 (0.40) CD274KCNH2GRIN2BGRM4TLR7
SCHEMBL21361259 0.79 CCR8 (0.47) KCNH2CCR8MAPT
SCHEMBL24120381 0.78 MAOB (0.39) KCNH2GRIN2BGRM4TLR7NPC1
SCHEMBL22859732 0.76 SLC6A9 (0.34) POLBMAPT
SCHEMBL21361231 0.76 TNKS2 (0.36) KCNH2GRIN2BGRM4NPC1
SCHEMBL24120382 0.75 GRM4 (0.38) CD274KCNH2GRIN2BGRM4TLR7
SCHEMBL24120432 0.74 RBP4 (0.41) KCNH2CCR8GRIN2BGRM4MAPT
SCHEMBL21361306 0.74 GAA (0.44) KCNH2CCR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019175117-A1 SPIRO CYCLOHEXANEDIONE DERIVATES AS HERBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2019-09-19 WO disclosed