SCHEMBL21362537

SCHEMBL21362537

COCc1ccc(C(=O)c2ccc(C)cc2Br)cc1F

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.37
NPC1 O15118 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
MAOB P27338 1/20 0.37
MAPK14 Q16539 10/20 0.37
ALDH1A1 P00352 1/20 0.35
KDM5A P29375 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
ROCK2 O75116 1/20 0.35
MAPK12 P53778 1/20 0.35
MAPK11 Q15759 1/20 0.35
STRADA Q7RTN6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20158084 0.81 HTT (0.54) MAPTNPC1MAPK1HTTALDH1A1
SCHEMBL20157484 0.78 ALDH1A1 (0.48) MAPTNPC1MAPK1HTTALDH1A1
SCHEMBL20157547 0.75 MAPT (0.50) MAPTNPC1MAPK1HTTALDH1A1
SCHEMBL12121014 0.74 IDO1 (0.42) MAPTMAOBMAPK14ALDH1A1KDM5A
SCHEMBL20157816 0.73 MAPT (0.51) MAPTNPC1MAPK1HTTALDH1A1
SCHEMBL11964298 0.73 HTT (0.57) MAPK1HTTMAOBKDM5AKDM4C
Sulfamide SCHEMBL21352056 0.73 ALDH1A1 (0.43) MAPTNPC1MAPK1HTTALDH1A1
Ammonia Solution, Strong SCHEMBL28443748 0.73 IDO1 (0.41) MAPTMAOBMAPK14ALDH1A1KDM5A
SCHEMBL20157414 0.73 NPC1 (0.58) MAPTNPC1MAPK1HTTALDH1A1
SCHEMBL20157483 0.72 ALDH1A1 (0.50) MAPTNPC1MAPK1HTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed