SCHEMBL21362791

SCHEMBL21362791

C=Cc1ccc(C(=O)c2ccc(C)cc2Br)cc1OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.44
CYP1A2 P05177 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
HPGD P15428 3/20 0.40
CYP2D6 P10635 1/20 0.40
ABL1 P00519 1/20 0.40
RIN1 Q13671 1/20 0.40
MAPT P10636 4/20 0.40
HTT P42858 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
SLC22A6 Q4U2R8 1/20 0.39
SLC22A8 Q8TCC7 1/20 0.39
NPC1 O15118 2/20 0.39
KMT2A Q03164 3/20 0.38
GAA P10253 2/20 0.38
MEN1 O00255 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21362533 0.85 ACHE (0.43) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL20157483 0.83 ALDH1A1 (0.50) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL21564805 0.81 ALDH1A1 (0.48) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL20157484 0.81 ALDH1A1 (0.48) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL20158084 0.78 HTT (0.54) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
Sulfamide SCHEMBL21352056 0.76 ALDH1A1 (0.43) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL20157414 0.76 NPC1 (0.58) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL20158021 0.75 LCK (0.46) ALDH1A1CYP1A2CYP2C19CYP2C9HPGD
SCHEMBL14678442 0.74 ACHE (0.56) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL29160653 0.73 CA12 (0.62) ALDH1A1CYP1A2CYP2C19CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed