SCHEMBL21363749

SCHEMBL21363749

C=CCc1cc2c(cc1NS(C)(=O)=O)OCO2

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.43
MAPT P10636 2/20 0.43
CYP1A2 P05177 1/20 0.43
PTGS1 P23219 1/20 0.43
PTGS2 P35354 1/20 0.43
PIK3CD O00329 1/20 0.40
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 1/20 0.39
RAB9A P51151 1/20 0.39
GLO1 Q04760 1/20 0.38
MEN1 O00255 1/20 0.38
PKM P14618 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
POLB P06746 3/20 0.36
MCHR1 Q99705 2/20 0.36
ALOX15 P16050 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21363755 0.73 MAPT (0.43) CYP3A4MAPTCYP1A2PTGS1PTGS2
SCHEMBL30860765 0.73 PTGS1 (0.44) MAPTPTGS1PTGS2PIK3CDALDH1A1
SCHEMBL11696893 0.71 CYP3A4 (0.53) CYP3A4MAPTCYP1A2ALDH1A1KDM4E
SCHEMBL7797624 0.71 CYP3A4 (0.53) CYP3A4MAPTCYP1A2ALDH1A1RAB9A
SCHEMBL8420054 0.70 KEAP1 (0.46) PTGS1ALDH1A1KDM4EKMT2AHPGD
SCHEMBL30860742 0.69 MAPT (0.51) CYP3A4MAPTCYP1A2PTGS1PTGS2
SCHEMBL21366573 0.69 NPC1 (0.54) CYP3A4MAPTCYP1A2PTGS2ALDH1A1
SCHEMBL21363792 0.69 MEN1 (0.44) CYP3A4MAPTCYP1A2ALDH1A1KDM4E
SCHEMBL1276635 0.69 CYP3A4 (0.55) CYP3A4MAPTCYP1A2ALDH1A1MEN1
SCHEMBL21363786 0.69 MAPT (0.48) CYP3A4MAPTCYP1A2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019175712-A1 NEW USES FOR CATECHOL MOLECULES AS INHIBITORS TO GLUTATHIONE S-TRANSFERASE METABOLIC PATHWAYS BASF CORPORATION (US) 2019-09-19 WO disclosed
WO-2019175713-A1 NEW CATECHOL MOLECULES AND THEIR USE AS INHIBITORS TO P450 RELATED METABOLIC PATHWAYS BASF CORPORATION (US) 2019-09-19 WO disclosed