SCHEMBL21367167

SCHEMBL21367167

OCn1ccc2c(Cl)ncnc21

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 1/20 0.44
FGFR1 P11362 2/20 0.44
FGFR4 P22455 2/20 0.44
NOTUM Q6P988 1/20 0.39
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
P2RX7 Q99572 2/20 0.35
FDPS P14324 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
KCNH2 Q12809 1/20 0.33
SCN5A Q14524 1/20 0.33
SCN9A Q15858 1/20 0.33
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4255524 0.82 SLC22A12 (0.41) SLC22A12FGFR1FGFR4NOTUMPDE4A
SCHEMBL28194794 0.81 SLC22A12 (0.42) SLC22A12FGFR1FGFR4NOTUMPDE4A
SCHEMBL4008337 0.80 NOTUM (0.47) SLC22A12FGFR1FGFR4NOTUMP2RX7
SCHEMBL21822975 0.79 ADORA2A (0.41) SLC22A12FGFR1FGFR4NOTUMPDE4A
SCHEMBL4015921 0.79 FGFR1 (0.40) SLC22A12FGFR1FGFR4NOTUMPDE4A
SCHEMBL19993789 0.79 ADK (0.45) PRMT5WDR77
SCHEMBL24753119 0.78 FGFR1 (0.44) SLC22A12FGFR1FGFR4NOTUMPDE4A
SCHEMBL22942935 0.78 FGFR1 (0.39) SLC22A12FGFR1FGFR4NOTUMPDE4A
SCHEMBL7664462 0.78 FGFR1 (0.46) SLC22A12FGFR1FGFR4NOTUMPDE4A
SCHEMBL3541053 0.78 NOTUM (0.58) FGFR1FGFR4NOTUMKCNH2SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019178368-A1 SELECTIVE INHIBITORS OF PROTEIN ARGININE METHYLTRANSFERASE 5 (PRMT5) PRELUDE THERAPEUTICS, INCORPORATED (US) 2019-09-19 WO disclosed