SCHEMBL21369912

SCHEMBL21369912

CC1(C)CCC(=O)c2ccc(OS(=O)C(F)(F)F)cc21

nearest known ligand 0.32

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.32
PGR P06401 3/20 0.32
RXRA P19793 1/20 0.32
RXRB P28702 1/20 0.32
RXRG P48443 1/20 0.32
HTT P42858 2/20 0.31
LMNA P02545 1/20 0.31
CRHBP P24387 1/20 0.31
CRHR2 Q13324 1/20 0.31
ALDH1A1 P00352 2/20 0.30
MALT1 Q9UDY8 1/20 0.30
CYP3A4 P08684 1/20 0.30
THRB P10828 1/20 0.30
MAPK1 P28482 1/20 0.30
KDM4E B2RXH2 1/20 0.30
PPARG P37231 1/20 0.30
PRNP P04156 1/20 0.30
PDK2 Q15119 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1807301 0.78 DRD2 (0.39) MAOBRXRARXRBRXRGPRNP
SCHEMBL1808153 0.78 KDM4E (0.49) HTTALDH1A1MALT1CYP3A4THRB
SCHEMBL8180939 0.73 MAOB (0.53) MAOB
SCHEMBL15717088 0.71 MALT1 (0.41) PGRMALT1
SCHEMBL24362396 0.71 KDM4E (0.59) MAOBHTTALDH1A1KDM4E
SCHEMBL5648628 0.70 PGR (0.49) MAOBPGRHTTALDH1A1CYP3A4
SCHEMBL24357642 0.69 KDM4E (0.50) MAOBHTTALDH1A1KDM4E
SCHEMBL24357847 0.69 MAOB (0.44) MAOBALDH1A1
SCHEMBL13613855 0.69 PGR (0.37) MAOBPGRRXRALMNAALDH1A1
SCHEMBL8648418 0.69 HPGD (0.43) PGRRXRARXRBRXRGLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2592071-B1 Tricyclic heterocyclic compounds BRISTOL MYERS SQUIBB CO (US) 2019-09-18 EP disclosed