SCHEMBL21371124

SCHEMBL21371124

Cc1cccc(Oc2ccc(Br)cc2C=O)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.51
ALDH1A1 P00352 4/20 0.45
GAA P10253 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
PTGDR2 Q9Y5Y4 1/20 0.44
LMNA P02545 5/20 0.42
KMT2A Q03164 2/20 0.42
AR P10275 1/20 0.42
MAPK1 P28482 1/20 0.42
ERN1 O75460 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ACHE P22303 1/20 0.40
HTT P42858 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
MAOB P27338 1/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2075254 0.83 LMNA (0.62) NPSR1ALDH1A1GAAL3MBTL1PTGDR2
SCHEMBL12438312 0.82 MAOB (0.45) NPSR1ALDH1A1GAAPTGDR2LMNA
SCHEMBL276480 0.79 EPAS1 (0.49) GAAPTGDR2LMNAKMT2AAR
SCHEMBL276011 0.78 PTGDR2 (0.46) NPSR1ALDH1A1L3MBTL1PTGDR2LMNA
SCHEMBL276112 0.78 PTGDR2 (0.46) NPSR1ALDH1A1GAAL3MBTL1PTGDR2
SCHEMBL275629 0.77 LMNA (0.61) NPSR1ALDH1A1GAAL3MBTL1PTGDR2
SCHEMBL1128457 0.77 AR (0.62) ALDH1A1GAAL3MBTL1ARMAPK1
SCHEMBL1643529 0.77 PTGDR2 (0.43) NPSR1ALDH1A1GAAPTGDR2LMNA
SCHEMBL5606306 0.77 ACHE (0.49) NPSR1ALDH1A1L3MBTL1PTGDR2LMNA
SCHEMBL21129706 0.76 LMNA (0.62) NPSR1ALDH1A1GAALMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019178480-A1 PYRAZOLE-CONTAINING MACROPHAGE MIGRATION INHIBITORY FACTOR INHIBITORS YALE UNIVERSITY (US) 2019-09-19 WO disclosed