SCHEMBL21371998

SCHEMBL21371998

Cn1ncc2ccc(SCC3CCC3)cc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 4/20 0.44
NOTUM Q6P988 1/20 0.38
CYP11B2 P19099 1/20 0.36
PTGER3 P43115 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2E1 P05181 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C8 P10632 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2B6 P20813 1/20 0.35
CYP2C19 P33261 1/20 0.35
GPR84 Q9NQS5 1/20 0.35
ALDH1A1 P00352 1/20 0.34
ERCC1 P07992 1/20 0.34
ERCC4 Q92889 1/20 0.34
PDE1C Q14123 1/20 0.34
CDK8 P49336 1/20 0.34
USP30 Q70CQ3 1/20 0.34
PFKFB3 Q16875 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24908252 0.75 NOTUM (0.43) ARNOTUMCYP11B2CYP1A2ERCC1
SCHEMBL16407110 0.69 ALDH1A1 (0.41) NOTUMCYP11B2CYP1A2ALDH1A1ERCC1
SCHEMBL29855932 0.68 HDAC4 (0.49) NOTUMCYP11B2PTGER3ERCC1ERCC4
SCHEMBL25702594 0.68 MAOB (0.51) CYP1A2CYP2E1CYP3A4CYP2C8CYP2D6
SCHEMBL30438880 0.68 MAOB (0.51) CYP1A2CYP2E1CYP3A4CYP2C8CYP2D6
SCHEMBL11586993 0.66 AR (0.49) ARCYP1A2CYP2E1CYP3A4CYP2C8
SCHEMBL21309298 0.66 HTR2A (0.35) NOTUMCYP11B2ERCC1ERCC4PDE1C
SCHEMBL20883607 0.65 AR (0.47) ARCYP11B2CYP1A2ALDH1A1PDE1C
SCHEMBL425168 0.65 KMO (0.57) NOTUMCYP11B2CYP1A2ERCC1ERCC4
SCHEMBL29901474 0.65 KMO (0.57) NOTUMCYP11B2CYP1A2ERCC1ERCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3180344-B1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES USEFUL FOR INHIBITING JANUS KINASE PFIZER (US) 2019-09-18 EP disclosed