SCHEMBL21372201

SCHEMBL21372201

Fc1cc(I)cc2c1OCCN2

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PIK3CD O00329 3/20 0.34
BTK Q06187 3/20 0.34
CDK4 P11802 1/20 0.34
CDK6 Q00534 1/20 0.34
AR P10275 1/20 0.34
EGFR P00533 1/20 0.33
FABP6 P51161 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2361983 0.81 ALDH1A1 (0.37) ALDH1A1GAAMAPTHSD17B10PIK3CD
SCHEMBL12116975 0.79 ALDH1A1 (0.50) ALDH1A1GAAMAPTHSD17B10PIK3CD
SCHEMBL13035938 0.79 ALDH1A1 (0.35) ALDH1A1GAAMAPTHSD17B10PIK3CD
SCHEMBL29620781 0.79 ALDH1A1 (0.35) ALDH1A1GAAMAPTHSD17B10PIK3CD
SCHEMBL25367179 0.76 AR (0.36) ALDH1A1GAAMAPTHSD17B10PIK3CD
SCHEMBL3329757 0.75 DHFR (0.34) ALDH1A1GAAMAPTHSD17B10PIK3CD
SCHEMBL13036607 0.75 ALDH1A1 (0.36) ALDH1A1GAAMAPTHSD17B10PIK3CD
SCHEMBL3328643 0.75 AR (0.35) ALDH1A1GAAMAPTHSD17B10PIK3CD
SCHEMBL16655910 0.75 PIK3CD (0.33) ALDH1A1GAAMAPTHSD17B10PIK3CD
SCHEMBL30284433 0.70 ADORA2A (0.43) ALDH1A1GAAMAPTHSD17B10PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3639824-A1 TRICYCLIC NITROGEN CONTAINING COMPOUNDS FOR TREATING NEISSERIA GONORRHOEA INFECTION GlaxoSmithKline Intellectual Property Development Limited (GB) 2020-04-22 EP disclosed
EP-3182973-B1 TRICYCLIC NITROGEN CONTAINING COMPOUNDS FOR TREATING NEISSERIA GONORRHOEA INFECTION GLAXOSMITHKLINE IP DEV LTD (GB) 2019-09-18 EP disclosed