2-Phenylthiazole

2-Phenylthiazole

SCHEMBL2137280

c1ccc(-c2nccs2)cc1.c1ccc2[nH]cnc2c1

nearest known ligand 0.64

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 2/20 0.64
QPCT Q16769 5/20 0.46
CYP2A6 P11509 1/20 0.45
RAB9A P51151 1/20 0.42
LOXL2 Q9Y4K0 1/20 0.41
METAP1 P53582 1/20 0.40
QPCTL Q9NXS2 2/20 0.40
ADRB2 P07550 1/20 0.39
PARP1 P09874 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
CDC7 O00311 1/20 0.38
KAT6A Q92794 1/20 0.38
KDR P35968 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Biphenyl SCHEMBL14655620 0.80 SMN1; SMN2 (0.48) PDPK1QPCTRAB9AQPCTLPARP1
2-Phenylthiazole SCHEMBL70646 0.80 PDPK1 (1.00) PDPK1CYP2A6RAB9ALOXL2METAP1
Benzimidazole SCHEMBL28095510 0.80 ALDH1A1 (0.50) PDPK1QPCTRAB9AQPCTLPARP1
SCHEMBL14720160 0.79 QPCT (0.48) PDPK1QPCTCYP2A6LOXL2QPCTL
2-Phenylthiazole SCHEMBL10519953 0.78 PDPK1 (0.95) PDPK1CYP2A6RAB9ALOXL2METAP1
2-Phenylthiazole SCHEMBL4939218 0.78 PDPK1 (0.95) PDPK1CYP2A6RAB9ALOXL2METAP1
2-Phenylthiazole SCHEMBL10667585 0.78 PDPK1 (0.95) PDPK1CYP2A6RAB9ALOXL2METAP1
2-Phenylthiazole SCHEMBL28319382 0.78 PDPK1 (0.95) PDPK1CYP2A6RAB9ALOXL2METAP1
2-Phenylthiazole SCHEMBL27882225 0.78 PDPK1 (0.95) PDPK1CYP2A6RAB9ALOXL2METAP1
Benzimidazole SCHEMBL1347288 0.78 KDM4E (0.50) PDPK1QPCTRAB9AQPCTLPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120101032-A1 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2012-04-26 US disclosed
WO-2012054874-A1 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2012-04-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120101032-A1 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION EIF2AK2, HAVCR2, EIF4A2 PDPK1 2409/4885QPCT 506/4885CYP2A6 227/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.