SCHEMBL21383210

SCHEMBL21383210

O=C(O)c1cnc2n[nH]cc2n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 4/20 0.49
ALDH1A1 P00352 2/20 0.49
HPGD P15428 1/20 0.49
HSD17B10 Q99714 1/20 0.49
AKR1B1 P15121 1/20 0.40
MGAM O43451 1/20 0.34
KDM4E B2RXH2 5/20 0.33
HCAR2 Q8TDS4 2/20 0.33
NAPRT Q6XQN6 1/20 0.33
CCNE2 O96020 2/20 0.33
CCNE1 P24864 2/20 0.33
CDK2 P24941 2/20 0.33
TSHR P16473 2/20 0.32
P4HA1 P13674 1/20 0.32
MIF P14174 1/20 0.32
P4HTM Q9NXG6 1/20 0.32
ACMSD Q8TDX5 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CCNB2 O95067 1/20 0.32
CDK1 P06493 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11865607 0.84 ALDH1A1 (0.33) ALOX15ALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL17608657 0.70 MGAM (0.48) ALOX15ALDH1A1HPGDHSD17B10MGAM
SCHEMBL21383793 0.69 CCNE2 (0.31) CCNE2CCNE1CDK2
SCHEMBL27158053 0.69 ALOX15 (0.50) ALOX15ALDH1A1HPGDHSD17B10AKR1B1
SCHEMBL6317502 0.69 ALOX15 (0.50) ALOX15ALDH1A1HPGDHSD17B10AKR1B1
SCHEMBL17443543 0.68 KDM4E (0.41) ALOX15ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL9903279 0.68 ALDH1A1 (0.49) ALOX15ALDH1A1HPGDHSD17B10AKR1B1
SCHEMBL30899548 0.68 ALOX15 (0.62) ALOX15ALDH1A1HPGDHSD17B10MGAM
SCHEMBL11617994 0.68 ALOX15 (0.62) ALOX15ALDH1A1HPGDHSD17B10MGAM
SCHEMBL5254858 0.68 KDM4E (0.41) ALOX15ALDH1A1HPGDHSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3768680-A1 PYRAZOLO[3,4-B]PYRAZINE SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF Relay Therapeutics, Inc. (US) 2021-01-27 EP disclosed
WO-2019183364-A1 PYRAZOLO[3,4-B]PYRAZINE SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed