SCHEMBL21383369

SCHEMBL21383369

Cn1nccc1NC(=O)CCl

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.55
POLB P06746 1/20 0.55
ALDH1A1 P00352 8/20 0.49
LMNA P02545 5/20 0.49
SMN1; SMN2 Q16637 4/20 0.49
HTT P42858 3/20 0.49
KDM4E B2RXH2 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
HSP90AA1 P07900 1/20 0.48
HSP90AB1 P08238 1/20 0.48
GAA P10253 3/20 0.45
EGFR P00533 1/20 0.42
NPC1 O15118 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
RAB9A P51151 1/20 0.42
OXTR P30559 1/20 0.42
AVPR1A P37288 1/20 0.42
JAK2 O60674 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29128621 0.87 KMT2A (0.57) KMT2APOLBALDH1A1LMNASMN1; SMN2
SCHEMBL26789473 0.84 POLB (0.59) KMT2APOLBALDH1A1KDM4EL3MBTL1
SCHEMBL12630078 0.80 POLB (0.52) KMT2APOLBALDH1A1KDM4EL3MBTL1
SCHEMBL30516912 0.79 POLB (0.51) KMT2APOLBLMNASMN1; SMN2HTT
SCHEMBL49946 0.78 KMT2A (0.57) KMT2APOLBALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL3268236 0.78 KMT2A (0.57) KMT2APOLBALDH1A1SMN1; SMN2HSP90AA1
SCHEMBL9523223 0.77 KMT2A (0.55) KMT2APOLBALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL1858809 0.76 POLB (0.51) KMT2APOLBLMNAL3MBTL1HSP90AA1
SCHEMBL1863466 0.75 POLB (0.48) KMT2APOLBLMNAHSP90AA1HSP90AB1
SCHEMBL2632922 0.75 KMT2A (0.62) KMT2APOLBALDH1A1SMN1; SMN2HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12157742-B2 Kinase inhibitors exhibiting anti-cancer activity and their method of use ALLCRON PHARMA INC. (US) 2024-12-03 US disclosed
US-20230399337-A1 NOVEL KINASE INHIBITORS EXHIBITING ANTI-CANCER ACTIVITY AND THEIR METHOD OF USE ALLCRON PHARMA INC. 2023-12-14 US disclosed
US-20230399337-A1 NOVEL KINASE INHIBITORS EXHIBITING ANTI-CANCER ACTIVITY AND THEIR METHOD OF USE ALLCRON PHARMA INC. 2023-12-14 US disclosed
US-20230399337-A1 NOVEL KINASE INHIBITORS EXHIBITING ANTI-CANCER ACTIVITY AND THEIR METHOD OF USE ALLCRON PHARMA INC. 2023-12-14 US disclosed
US-11697654-B2 Kinase inhibitors exhibiting anti-cancer activity and their method of use ALLCRON PHARMA INC. (US) 2023-07-11 US disclosed
US-11697654-B2 Kinase inhibitors exhibiting anti-cancer activity and their method of use ALLCRON PHARMA INC. (US) 2023-07-11 US disclosed
US-11697654-B2 Kinase inhibitors exhibiting anti-cancer activity and their method of use ALLCRON PHARMA INC. (US) 2023-07-11 US disclosed
EP-3768682-B1 2-({2H,3H-[1,4]DIOXINO[2,3-G]QUINOLIN-7-YL}SULFANYL)ACETAMIDE DERIVATIVES AS BCR-ABL KINASE INHIBITORS FOR THE TREATMENT OF CANCER ALLCRON PHARMA INC (US) 2023-07-05 EP disclosed
EP-3768682-B1 2-({2H,3H-[1,4]DIOXINO[2,3-G]QUINOLIN-7-YL}SULFANYL)ACETAMIDE DERIVATIVES AS BCR-ABL KINASE INHIBITORS FOR THE TREATMENT OF CANCER ALLCRON PHARMA INC (US) 2023-07-05 EP disclosed
US-20210040104-A1 NOVEL KINASE INHIBITORS EXHIBITING ANTI-CANCER ACTIVITY AND THEIR METHOD OF USE ALLCRON PHARMA INC. 2021-02-11 US disclosed
US-20210040104-A1 NOVEL KINASE INHIBITORS EXHIBITING ANTI-CANCER ACTIVITY AND THEIR METHOD OF USE ALLCRON PHARMA INC. 2021-02-11 US disclosed
EP-3768682-A1 NOVEL KINASE INHIBITORS EXHIBITING ANTI-CANCER ACTIVITY AND THEIR METHOD OF USE Allcron Pharma Inc. (US) 2021-01-27 EP disclosed
WO-2019182944-A1 NOVEL KINASE INHIBITORS EXHIBITING ANTI-CANCER ACTIVITY AND THEIR METHOD OF USE ALLCRON PHARMA INC. (US) 2019-09-26 WO disclosed
WO-2019182944-A1 NOVEL KINASE INHIBITORS EXHIBITING ANTI-CANCER ACTIVITY AND THEIR METHOD OF USE ALLCRON PHARMA INC. (US) 2019-09-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210040104-A1 NOVEL KINASE INHIBITORS EXHIBITING ANTI-CANCER ACTIVITY AND THEIR METHOD OF USE ABL1, MCL1, ABL2 KMT2A 370/4885POLB 3176/4885ALDH1A1 3210/4885
US-20230399337-A1 NOVEL KINASE INHIBITORS EXHIBITING ANTI-CANCER ACTIVITY AND THEIR METHOD OF USE ABL1, MCL1, ABL2 KMT2A 370/4885POLB 3176/4885ALDH1A1 3210/4885
US-11697654-B2 Kinase inhibitors exhibiting anti-cancer activity and their method of use ABL1, MCL1, ABL2 KMT2A 358/4885POLB 2592/4885ALDH1A1 2686/4885
US-12157742-B2 Kinase inhibitors exhibiting anti-cancer activity and their method of use ABL1, MCL1, ABL2 KMT2A 358/4885POLB 2592/4885ALDH1A1 2686/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.