SCHEMBL21385166

SCHEMBL21385166

COc1ccc(N2CCC(C(C)NC(=O)N=[N+]=[N-])CC2)cn1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.42
CHRNA4 P43681 3/20 0.42
CHRNB4 P30926 2/20 0.42
CHRNA3 P32297 2/20 0.42
ACACB O00763 10/20 0.41
OGA O60502 1/20 0.40
PIK3CG P48736 1/20 0.39
HRH3 Q9Y5N1 1/20 0.38
F10 P00742 1/20 0.37
SMYD3 Q9H7B4 1/20 0.37
LCAT P04180 1/20 0.37
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30574427 1.00 CHRNB2 (0.42) CHRNB2CHRNA4CHRNB4CHRNA3ACACB
SCHEMBL21384602 0.84 ACACB (0.44) ACACBSMYD3
SCHEMBL28455935 0.80 SMYD3 (0.42) ACACBSMYD3
SCHEMBL21384592 0.76 CHRNB2 (0.50) CHRNB2CHRNA4CHRNB4CHRNA3ACACB
SCHEMBL30574420 0.76 CHRNB2 (0.50) CHRNB2CHRNA4CHRNB4CHRNA3ACACB
SCHEMBL21384587 0.73 CHRNB2 (0.47) CHRNB2CHRNA4CHRNB4CHRNA3ACACB
SCHEMBL21384594 0.72 GAA (0.43) ACACB
Hydrochloric Acid SCHEMBL30574425 0.72 CHRNB2 (0.53) CHRNB2CHRNA4CHRNB4CHRNA3ACACB
Hydrochloric Acid SCHEMBL21384628 0.72 CHRNB2 (0.53) CHRNB2CHRNA4CHRNB4CHRNA3ACACB
SCHEMBL21396932 0.72 F10 (0.39) CHRNB2CHRNA4CHRNB4CHRNA3ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117185987-A Amidine and guanidine derivatives, preparation method and medical application thereof 四川科伦博泰生物医药股份有限公司 2023-12-08 CN disclosed
CN-111630048-B Amidine and guanidine derivatives, preparation method and medical application thereof 四川科伦博泰生物医药股份有限公司 2023-09-29 CN disclosed
CN-111630048-A Amidine and guanidine derivatives, preparation method and application thereof in medicines 四川科伦博泰生物医药股份有限公司 2020-09-04 CN disclosed
WO-2019179362-A1 AMIDINE AND GUANIDINE DERIVATIVES, PREPARATION METHOD THEREFOR AND MEDICAL USES THEREOF 四川科伦博泰生物医药股份有限公司 2019-09-26 WO disclosed
WO-2019179362-A1 AMIDINE AND GUANIDINE DERIVATIVES, PREPARATION METHOD THEREFOR AND MEDICAL USES THEREOF 四川科伦博泰生物医药股份有限公司 2019-09-26 WO disclosed