SCHEMBL21386776

SCHEMBL21386776

C=CC(=O)N1CCC[C@@H](Nc2ncnc(N)c2C(=N)c2ccc(Oc3c(F)cccc3F)nc2F)C1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BTK Q06187 13/20 0.57
EGFR P00533 4/20 0.52
JAK3 P52333 5/20 0.50
JAK1 P23458 1/20 0.47
ITK Q08881 2/20 0.46
BLK P51451 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21386772 0.96 BTK (0.51) BTKEGFRJAK3JAK1ITK
SCHEMBL21386763 0.92 BTK (0.58) BTKEGFRJAK3JAK1ITK
SCHEMBL21386703 0.92 BTK (0.58) BTKEGFRJAK3JAK1ITK
SCHEMBL21386783 0.91 BTK (0.67) BTKEGFRJAK3JAK1BLK
SCHEMBL21386788 0.89 BTK (0.59) BTKEGFRJAK3JAK1ITK
SCHEMBL21386736 0.88 BTK (0.61) BTKEGFRJAK3JAK1ITK
SCHEMBL21386773 0.88 BTK (0.52) BTKEGFRJAK3ITKBLK
SCHEMBL21386655 0.87 BTK (0.60) BTKEGFRITKBLK
SCHEMBL21386725 0.83 BTK (0.67) BTKEGFRJAK3JAK1ITK
SCHEMBL21386778 0.81 BTK (0.66) BTKEGFRJAK3JAK1ITK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3543239-A1 SELECTIVE BRUTON'S TYROSINE KINASE INHIBITOR AND USE THEREOF Hangzhou Hertz Pharmaceutical Co., Ltd. (CN) 2019-09-25 EP disclosed