SCHEMBL21387637

SCHEMBL21387637

CC(C)(C=O)c1ccnc(NS(C)(=O)=O)n1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.45
CTPS1 P17812 8/20 0.44
NPSR1 Q6W5P4 1/20 0.39
SYK P43405 4/20 0.39
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38
MAPK8 P45983 1/20 0.37
MAPK10 P53779 1/20 0.37
ALDH1A1 P00352 1/20 0.35
AR P10275 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21387725 0.85 CTPS1 (0.44) MAPK1CTPS1NPSR1SYKMAPT
SCHEMBL21387640 0.82 CTPS1 (0.52) CTPS1
SCHEMBL21387680 0.81 CTPS1 (0.46) MAPK1CTPS1NPSR1MAPTCYP2C9
SCHEMBL21373740 0.75 CTPS1 (0.52) MAPK1CTPS1
SCHEMBL21387600 0.72 CTPS1 (0.31) CTPS1SYK
SCHEMBL12522323 0.72 MAPK1 (0.69) MAPK1NPSR1MAPTCYP2C9ALDH1A1
SCHEMBL21387688 0.71 SYK (0.32) SYK
SCHEMBL9182494 0.70 MAPK1 (0.48) MAPK1CTPS1NPSR1MAPTCYP2C9
SCHEMBL30059838 0.70 MAPK1 (0.48) MAPK1CTPS1NPSR1MAPTCYP2C9
SCHEMBL21392313 0.68 CTPS1 (0.44) MAPK1CTPS1SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3543232-A1 AMINOPYRIMIDINE DERIVATIVES AS CTPS1 INHIBITORS Step Pharma S.A.S. (FR) 2019-09-25 EP disclosed