SCHEMBL21387680

SCHEMBL21387680

CC(C)(C=O)c1ccnc(NS(=O)(=O)C2(C)CC2)n1

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTPS1 P17812 12/20 0.46
NPSR1 Q6W5P4 1/20 0.35
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21387637 0.81 MAPK1 (0.45) CTPS1NPSR1MAPTCYP2C9MAPK1
SCHEMBL21373711 0.79 CTPS1 (0.54) CTPS1
SCHEMBL21387725 0.79 CTPS1 (0.44) CTPS1NPSR1MAPTCYP2C9MAPK1
SCHEMBL21387640 0.78 CTPS1 (0.52) CTPS1
SCHEMBL21387688 0.75 SYK (0.32)
SCHEMBL21387600 0.69 CTPS1 (0.31) CTPS1
SCHEMBL22758565 0.69 CTPS1 (0.37) CTPS1NPSR1MAPTCYP2C9
SCHEMBL21392095 0.63 CTPS1 (0.50) CTPS1
Hydrochloric Acid SCHEMBL21384760 0.62 CTPS1 (0.49) CTPS1
SCHEMBL23173845 0.61 TSHR (0.54) MAPK1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3543232-A1 AMINOPYRIMIDINE DERIVATIVES AS CTPS1 INHIBITORS Step Pharma S.A.S. (FR) 2019-09-25 EP disclosed