SCHEMBL21387928

SCHEMBL21387928

COc1ccc(CO[C@@H]2OCC(O[Si](C)(C)C(C)(C)C)[C@H](N)C2OC(C)=O)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
CYP2D6 P10635 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
CYP2C19 P33261 2/20 0.37
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37
HIF1A Q16665 1/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP2C9 P11712 1/20 0.37
KMT2A Q03164 1/20 0.37
SLC2A1 P11166 1/20 0.37
PREP P48147 2/20 0.33
IDO1 P14902 2/20 0.32
AGXT P21549 2/20 0.32
GJB2 P29033 1/20 0.32
GJA1 P17302 1/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21387868 1.00 CA1 (0.39) CA1CA2CA9CYP2D6SMN1; SMN2
SCHEMBL21387904 0.84 GJB2 (0.38) CYP2C19IDO1AGXTGJB2GJA1
SCHEMBL17472212 0.84 CYP2D6 (0.34) CA1CA2CA9CYP2D6SMN1; SMN2
SCHEMBL21387848 0.72 CYP3A4 (0.32) CYP3A4
SCHEMBL17472164 0.72
SCHEMBL21387847 0.72
SCHEMBL17274148 0.70 CYP2D6 (0.33) CYP2D6SMN1; SMN2CYP2C19LMNAMAPK1
SCHEMBL17472165 0.70 CYP2D6 (0.33) CYP2D6SMN1; SMN2CYP2C19LMNAMAPK1
SCHEMBL7150003 0.68 CA1 (0.52) CA1CA2CA9LMNAALDH1A1
SCHEMBL7150000 0.68 CA1 (0.52) CA1CA2CA9LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3142672-B1 AMPHOTERICIN B DERIVATIVE WITH REDUCED TOXICITY UNIV ILLINOIS (US) 2019-09-25 EP disclosed