SCHEMBL21387904

SCHEMBL21387904

COc1ccc(COC2OCC(O[Si](C)(C)C(C)(C)C)[C@H](N)[C@H]2O)cc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GJB2 P29033 1/20 0.38
GJA1 P17302 1/20 0.38
IDO1 P14902 2/20 0.36
AGXT P21549 2/20 0.36
THRB P10828 1/20 0.32
TACR1 P25103 1/20 0.32
NAAA Q02083 1/20 0.32
SLC5A1 P13866 1/20 0.31
SLC5A2 P31639 1/20 0.31
REN P00797 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
MAOB P27338 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21387868 0.84 CA1 (0.39) GJB2GJA1IDO1AGXTTHRB
SCHEMBL21387928 0.84 CA1 (0.39) GJB2GJA1IDO1AGXTTHRB
SCHEMBL17472164 0.82
SCHEMBL15032442 0.73 NAAA (0.38) IDO1AGXTTHRBNAAAREN
SCHEMBL17472212 0.72 CYP2D6 (0.34) CYP2C19
SCHEMBL22639406 0.72 THRB (0.35) IDO1AGXTTHRBTACR1NAAA
SCHEMBL29773823 0.70 NAAA (0.44) IDO1AGXTTHRBNAAAKDM4E
SCHEMBL16155041 0.69 IDO1 (0.36) IDO1AGXTTHRBTACR1NAAA
SCHEMBL24894254 0.69 KDM4E (0.32) IDO1AGXTTHRBRENKDM4E
SCHEMBL14363012 0.69 SLC6A2 (0.43) GJB2GJA1THRBTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3142672-B1 AMPHOTERICIN B DERIVATIVE WITH REDUCED TOXICITY UNIV ILLINOIS (US) 2019-09-25 EP disclosed