SCHEMBL21390842

SCHEMBL21390842

CC(C)(CC(=O)CCCCc1nc2ccc(C(C)(C)O)cc2n1C1CCC1)CC(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 7/20 0.36
CYP11B2 P19099 5/20 0.35
CYP11B1 P15538 4/20 0.35
CYP19A1 P11511 2/20 0.35
ADRB1 P08588 1/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
RORC P51449 1/20 0.34
USP2 O75604 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ACSS2 Q9NR19 1/20 0.31
ALK Q9UM73 2/20 0.31
NTRK1 P04629 1/20 0.31
INSR P06213 1/20 0.31
LCK P06239 1/20 0.31
LTK P29376 1/20 0.31
AXL P30530 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21391106 0.87 HDAC1 (0.37) HDAC1CYP11B2CYP11B1CYP19A1ADRB1
SCHEMBL21390843 0.85 CYP19A1 (0.33) HDAC1CYP11B2CYP11B1CYP19A1
SCHEMBL21390845 0.85 HDAC1 (0.40) HDAC1CYP11B2CYP11B1CYP19A1ADRB1
SCHEMBL21390840 0.84 HDAC1 (0.35) HDAC1CYP11B2CYP11B1CYP19A1ADRB1
SCHEMBL21390841 0.83 HDAC1 (0.35) HDAC1CYP11B2CYP11B1CYP19A1ADRB1
SCHEMBL21391026 0.80 HDAC1 (0.37) HDAC1CYP11B2CYP11B1CYP19A1ADRB1
SCHEMBL18791675 0.79 EGFR (0.42) CYP11B2CYP11B1CYP19A1ADRB1ADRA2A
SCHEMBL23132031 0.79 CYP11B2 (0.41) HDAC1CYP11B2CYP11B1CYP19A1ADRB1
SCHEMBL21390674 0.77 ALK (0.37) HDAC1CYP11B2CYP11B1CYP19A1ADRB1
SCHEMBL21391041 0.77 HDAC1 (0.36) HDAC1CYP11B2CYP11B1CYP19A1ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019183148-A1 KV7 CHANNEL ACTIVATORS COMPOSITIONS AND METHODS OF USE KNOPP BIOSCIENCES LLC (US) 2019-09-26 WO disclosed