SCHEMBL21391039

SCHEMBL21391039

N#Cc1ccc2c(c1)CCCC/C=N\2

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.39
DRD2 P14416 2/20 0.39
DRD3 P35462 2/20 0.39
PNMT P11086 1/20 0.39
KDM1A O60341 2/20 0.38
CYP11B2 P19099 5/20 0.37
CYP19A1 P11511 6/20 0.36
CYP11B1 P15538 4/20 0.36
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
HDAC1 Q13547 2/20 0.33
HDAC8 Q9BY41 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
CXCR5 P32302 1/20 0.32
MAOA P21397 3/20 0.32
MAOB P27338 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28039609 0.88 PNMT (0.42) TRPA1DRD2DRD3PNMTKDM1A
SCHEMBL11017385 0.78 TRPA1 (0.44) TRPA1DRD2DRD3PNMTKDM1A
SCHEMBL24375978 0.75
SCHEMBL29741121 0.73 PNMT (0.60) DRD2DRD3PNMTKDM1ACYP11B2
SCHEMBL3363261 0.73 PNMT (0.60) DRD2DRD3PNMTKDM1ACYP11B2
Hydrochloric Acid SCHEMBL15205820 0.71 PNMT (0.58) DRD2DRD3PNMTKDM1ACYP11B2
SCHEMBL17350029 0.71 PNMT (0.58) DRD2DRD3PNMTKDM1ACYP11B2
SCHEMBL7647780 0.70 PNMT (0.44) TRPA1DRD2DRD3PNMTKDM1A
SCHEMBL12471274 0.70 TSHR (0.48) TRPA1NOS3NOS1NOS2MAOA
SCHEMBL8222195 0.69 PNMT (0.60) DRD2DRD3PNMTKDM1ACYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019183148-A1 KV7 CHANNEL ACTIVATORS COMPOSITIONS AND METHODS OF USE KNOPP BIOSCIENCES LLC (US) 2019-09-26 WO disclosed