SCHEMBL21392312

SCHEMBL21392312

COC(=O)C(C=O)c1cc(C(F)(F)F)nc(Cl)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.38
CYP2C19 P33261 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35
FFAR2 O15552 1/20 0.33
IGF1R P08069 3/20 0.32
MAPT P10636 2/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
KMT2A Q03164 1/20 0.32
ATF1 P18846 2/20 0.32
NFKB1 P19838 2/20 0.32
MRGPRX4 Q96LA9 1/20 0.31
SMARCA2 P51531 1/20 0.31
SMARCA4 P51532 1/20 0.31
SDHB P21912 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21381568 0.80 MAPK1 (0.44) MAPK1CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL21392136 0.77 LMNA (0.45) MAPK1CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL22767093 0.70 CYP2C19 (0.61) CYP2C19CYP3A4CYP2D6TSHRCRHBP
SCHEMBL16095194 0.70 MAPT (0.46) MAPTALDH1A1HPGDMRGPRX4SDHB
SCHEMBL22924876 0.69 IGF1R (0.36) MAPK1IGF1RMAPTALDH1A1HPGD
SCHEMBL5998172 0.68 PTGS1 (0.39) MAPK1CYP2C19CYP3A4CYP2D6TSHR
SCHEMBL21392139 0.67 KDM4E (0.47) MAPTMEN1ALDH1A1HPGDKMT2A
SCHEMBL30261798 0.66 KMO (0.45) TSHRIGF1RMAPTMEN1HPGD
SCHEMBL25859898 0.66 KMO (0.45) TSHRIGF1RMAPTMEN1HPGD
SCHEMBL6468496 0.65 NT5E (0.42) CYP2C19CYP3A4CYP2D6TSHRCRHBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019179652-A1 AMINOPYRIMIDINE DERIVATIVES AS CTPS1 INHIBITORS STEP PHARMA S.A.S. (FR) 2019-09-26 WO disclosed