SCHEMBL21393376

SCHEMBL21393376

C=C(OC)c1c(C)cncc1N

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GLA P06280 1/20 0.35
GAA P10253 1/20 0.35
ATM Q13315 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20187436 0.78 ALDH1A1 (0.50) KDM4EALDH1A1GLAGAAATM
SCHEMBL26151369 0.71 TDP1 (0.41) KDM4EALDH1A1GLAGAA
SCHEMBL18171007 0.71 KDM4E (0.43) KDM4EALDH1A1GLAGAA
SCHEMBL22490108 0.68
SCHEMBL20203202 0.67 MEN1 (0.37) KDM4EALDH1A1GLAGAA
SCHEMBL27365834 0.66
SCHEMBL19616148 0.66 AGXT (0.39) KDM4EALDH1A1GLAGAA
SCHEMBL22827595 0.64 ALDH1A1 (0.37) ALDH1A1GAA
SCHEMBL12915143 0.64
SCHEMBL541849 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019182925-A1 OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS GENENTECH, INC. (US) 2019-09-26 WO disclosed