SCHEMBL21393631

SCHEMBL21393631

C/C(N)=C(\C)c1c(N)nc[nH]c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GDA Q9Y2T3 1/20 0.43
PARP1 P09874 8/20 0.38
ALDH1A1 P00352 2/20 0.38
SLC2A1 P11166 1/20 0.37
KDM4E B2RXH2 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.34
PDPK1 O15530 1/20 0.34
CA12 O43570 1/20 0.34
ALOX15 P16050 1/20 0.34
CA9 Q16790 1/20 0.34
TNKS2 Q9H2K2 1/20 0.34
PIM1 P11309 2/20 0.34
BCL2 P10415 1/20 0.34
MCL1 Q07820 1/20 0.34
CHEK1 O14757 1/20 0.34
RPS6KA3 P51812 1/20 0.34
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26049473 0.69
SCHEMBL3170605 0.69
SCHEMBL4455591 0.68
SCHEMBL29812517 0.67 GDA (0.41) GDAPARP1ALDH1A1SLC2A1KDM4E
SCHEMBL11901381 0.67 GDA (0.44) GDAALDH1A1SLC2A1KDM4EGLA
SCHEMBL2942472 0.64 IP6K1 (0.41) GDAPARP1ALDH1A1KDM4EGLA
SCHEMBL29289348 0.64 GDA (0.42) GDAPARP1ALDH1A1SLC2A1KDM4E
SCHEMBL27660603 0.64 ALDH1A1 (0.39) GDAPARP1ALDH1A1KDM4EGLA
SCHEMBL14113725 0.63 ALDH1A1 (0.38) PARP1ALDH1A1SLC2A1PDPK1PIM1
SCHEMBL9918618 0.63 GDA (0.41) GDAPARP1ALDH1A1KDM4EGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019182925-A1 OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS GENENTECH, INC. (US) 2019-09-26 WO disclosed