SCHEMBL21393780

SCHEMBL21393780

C=Nc1c(Cl)ncc(C)c1C=O

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
RECQL P46063 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22716205 0.73 KDM4E (0.33) CYP1A2CYP3A4CYP2D6CYP2C19KDM4E
SCHEMBL22729409 0.72 KDM4E (0.38) CYP1A2CYP3A4CYP2D6CYP2C19KDM4E
SCHEMBL30082527 0.72 KDM4E (0.38) CYP1A2CYP3A4CYP2D6CYP2C19KDM4E
SCHEMBL21393415 0.71 ALDH1A1 (0.32)
SCHEMBL22715564 0.67 PIK3C3 (0.33) CYP3A4KDM4EMAPTRECQLNPSR1
SCHEMBL1044209 0.66 ALDH1A1 (0.35) CYP3A4KDM4EMAPTRECQLNPSR1
SCHEMBL20203314 0.66
SCHEMBL21393347 0.64
Pyridine SCHEMBL21226522 0.63 KDM4E (0.35) KDM4EMAPTRECQLNPSR1
SCHEMBL6920756 0.62 MEN1 (0.38) CYP1A2CYP3A4CYP2D6CYP2C19KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019182925-A1 OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS GENENTECH, INC. (US) 2019-09-26 WO disclosed