SCHEMBL21393826

SCHEMBL21393826

Cc1cnn2ncn(C)c(=O)c12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 10/20 0.34
NFE2L2 Q16236 1/20 0.33
ALDH1A1 P00352 3/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.31
XBP1 P17861 1/20 0.31
HTT P42858 1/20 0.31
RAB9A P51151 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
PIK3CD O00329 1/20 0.31
POLB P06746 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
CNR1 P21554 1/20 0.31
ACHE P22303 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA2B P29275 1/20 0.31
ADORA1 P30542 1/20 0.31
NTSR1 P30989 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25165834 0.77 TRPA1 (0.42) TRPA1ALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL21363445 0.77 TRPA1 (0.33) TRPA1ALDH1A1SMN1; SMN2KMT2AHPGD
SCHEMBL24375561 0.69 CYP1A2 (0.31) ALDH1A1SMN1; SMN2POLBKDM4EGLA
SCHEMBL17163966 0.65 HTT (0.36) ALDH1A1HTT
SCHEMBL8404472 0.64
SCHEMBL20203175 0.64 TRPA1 (0.41) TRPA1PIK3CDPOLBADORA3CNR1
SCHEMBL15382212 0.64 ALDH1A1 (0.33) ALDH1A1ADORA2AADORA2BF2KMT2A
SCHEMBL21895459 0.63 ADORA2A (0.35) ALDH1A1NPC1MAPTHTTRAB9A
SCHEMBL23679319 0.63 BRD9 (0.32) NFE2L2ALDH1A1MAPTRXFP1F2
SCHEMBL21363426 0.62 TRPA1 (0.36) TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019182925-A1 OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS GENENTECH, INC. (US) 2019-09-26 WO disclosed