SCHEMBL21394732

SCHEMBL21394732

N#Cc1cc(C(=O)Nc2ccc(Cc3ccc(F)c(F)c3)cn2)ccn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 4/20 0.48
KCNQ2 O43526 4/20 0.48
WNT1 P04628 1/20 0.44
GSK3B P49841 1/20 0.44
DYRK1A Q13627 1/20 0.44
MAOB P27338 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.41
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
ALDH1A1 P00352 1/20 0.40
PKM P14618 1/20 0.40
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CHEK1 O14757 1/20 0.40
CYP3A4 P08684 1/20 0.39
SCD O00767 1/20 0.39
PARP1 P09874 1/20 0.39
KMT2A Q03164 2/20 0.38
F10 P00742 1/20 0.38
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21394997 0.86 KCNQ3 (0.57) KCNQ3KCNQ2MAOBSIRT2NPC1
SCHEMBL21395118 0.84 KCNQ3 (0.43) KCNQ3KCNQ2MAOBSIRT2NPC1
SCHEMBL21395019 0.83 PARP1 (0.53) KCNQ3KCNQ2MAOBNPC1RAB9A
SCHEMBL21395146 0.82 KCNQ3 (0.44) KCNQ3KCNQ2SIRT2NPC1RAB9A
SCHEMBL21395078 0.82 CHEK1 (0.48) KCNQ3KCNQ2SIRT2NPC1RAB9A
SCHEMBL21394650 0.81 PARP1 (0.41) KCNQ3KCNQ2MAOBNPC1RAB9A
SCHEMBL21395010 0.80 TMPRSS4 (0.44) KCNQ3KCNQ2SIRT2NPC1RAB9A
SCHEMBL21394718 0.75 NPC1 (0.42) KCNQ3KCNQ2GSK3BMAOBSIRT2
SCHEMBL21394396 0.74 KCNQ3 (0.47) KCNQ3KCNQ2ALDH1A1
SCHEMBL21394712 0.74 PPARG (0.41) KCNQ3KCNQ2MAOBNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020198026-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-10-01 WO disclosed
WO-2019183587-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed