SCHEMBL21394976

SCHEMBL21394976

Cn1cc(C(=O)Nc2ccc(Cc3cncc(F)c3)cn2)ccc1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.41
CREBBP Q92793 1/20 0.40
CYP11B1 P15538 2/20 0.40
CYP11B2 P19099 2/20 0.40
DEGS1 O15121 1/20 0.40
CYP3A4 P08684 2/20 0.39
RXFP1 Q9HBX9 1/20 0.39
GCK P35557 2/20 0.38
NTRK1 P04629 1/20 0.38
WNT1 P04628 1/20 0.38
CLK2 P49760 1/20 0.38
CLK3 P49761 1/20 0.38
GSK3B P49841 1/20 0.38
DYRK1A Q13627 1/20 0.38
PARP1 P09874 1/20 0.38
F10 P00742 1/20 0.38
SLC6A3 Q01959 2/20 0.37
ALOX5 P09917 1/20 0.37
TBXAS1 P24557 1/20 0.37
EPHX2 P34913 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29356925 0.91 GCK (0.44) KDM4ECREBBPDEGS1RXFP1GCK
SCHEMBL21394784 0.91 GCK (0.44) KDM4ECREBBPDEGS1RXFP1GCK
SCHEMBL21395178 0.89 CYP11B1 (0.51) KDM4ECREBBPCYP11B1CYP11B2DEGS1
SCHEMBL29353782 0.89 KDM4E (0.51) KDM4ECREBBPDEGS1RXFP1GCK
SCHEMBL21394550 0.89 KDM4E (0.51) KDM4ECREBBPDEGS1RXFP1GCK
SCHEMBL21394636 0.88 F10 (0.43) CREBBPDEGS1CYP3A4F10ALDH1A1
SCHEMBL29356936 0.88 NPC1 (0.46) KDM4ECREBBPDEGS1GCKNTRK1
SCHEMBL21394601 0.88 NPC1 (0.46) KDM4ECREBBPDEGS1GCKNTRK1
SCHEMBL21394480 0.86 MAPT (0.44) KDM4ECREBBPDEGS1RXFP1GCK
SCHEMBL21384385 0.86 CREBBP (0.42) KDM4ECREBBPDEGS1RXFP1GCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020198026-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-10-01 WO disclosed
WO-2019183587-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed