SCHEMBL21395031

SCHEMBL21395031

N#Cc1cnc(C(=O)Nc2ccc(Cc3cc(F)cc(Cl)c3)cn2)cn1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 13/20 0.41
CYP3A4 P08684 1/20 0.40
GRM2 Q14416 1/20 0.40
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
PKM P14618 1/20 0.39
TSHR P16473 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TMPRSS4 Q9NRS4 1/20 0.39
SIRT2 Q8IXJ6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21394932 0.94 CHEK1 (0.42) CHEK1GRM2
SCHEMBL21395016 0.90 CHEK1 (0.40) CHEK1CYP3A4GRM2TMPRSS4SIRT2
SCHEMBL21395150 0.89 TMPRSS4 (0.43) CHEK1CYP3A4NPC1TSHRRAB9A
SCHEMBL21395032 0.89 SMN1; SMN2 (0.42) CYP3A4NPC1ALDH1A1PKMTSHR
SCHEMBL21395078 0.87 CHEK1 (0.48) CHEK1GRM2NPC1RAB9ASMN1; SMN2
SCHEMBL21395011 0.85 GRM4 (0.43) CHEK1GRM2TMPRSS4SIRT2
SCHEMBL21395002 0.84 TMPRSS4 (0.41) CYP3A4NPC1ALDH1A1PKMTSHR
SCHEMBL21394947 0.83 JUN (0.43) NPC1ALDH1A1PKMTSHRRAB9A
SCHEMBL21395154 0.82 TMPRSS4 (0.44) CYP3A4TMPRSS4SIRT2
SCHEMBL21394950 0.82 CHEK1 (0.49) CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020198026-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-10-01 WO disclosed
WO-2019183587-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed