SCHEMBL21397263

SCHEMBL21397263

COc1ccc(N2CCC(NC(=O)OC(C)(C)C)CC2)c(F)c1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.48
CKS1B P61024 1/20 0.46
SKP1 P63208 1/20 0.46
SKP2 Q13309 1/20 0.46
ALDH1A1 P00352 1/20 0.46
DRD2 P14416 3/20 0.45
DRD3 P35462 2/20 0.44
SUV39H2 Q9H5I1 2/20 0.43
PIK3CA P42336 1/20 0.43
MTOR P42345 1/20 0.43
PRKDC P78527 1/20 0.43
BTK Q06187 1/20 0.42
KCNA3 P22001 1/20 0.42
PIM1 P11309 1/20 0.42
PIM3 Q86V86 1/20 0.42
PIM2 Q9P1W9 1/20 0.42
CTSK P43235 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4435954 0.86 ALDH1A1 (0.47) CKS1BSKP1SKP2ALDH1A1DRD2
SCHEMBL15759214 0.86 CKS1B (0.47) ACACBCKS1BSKP1SKP2DRD2
SCHEMBL3212610 0.86 CKS1B (0.47) CKS1BSKP1SKP2ALDH1A1DRD2
SCHEMBL30783037 0.86 CKS1B (0.47) CKS1BSKP1SKP2ALDH1A1DRD2
SCHEMBL31653702 0.85 CKS1B (0.47) CKS1BSKP1SKP2ALDH1A1DRD2
SCHEMBL13229631 0.85 CKS1B (0.47) CKS1BSKP1SKP2DRD2DRD3
SCHEMBL10264448 0.83 DRD2 (0.48) CKS1BSKP1SKP2DRD2DRD3
SCHEMBL4439231 0.83 MAPT (0.55) ALDH1A1
SCHEMBL31318667 0.82 SUV39H2 (0.51) DRD2SUV39H2PIM1PIM3PIM2
SCHEMBL17557723 0.82 MAPT (0.56) CKS1BSKP1SKP2ALDH1A1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019179362-A1 AMIDINE AND GUANIDINE DERIVATIVES, PREPARATION METHOD THEREFOR AND MEDICAL USES THEREOF 四川科伦博泰生物医药股份有限公司 2019-09-26 WO disclosed