SCHEMBL21397973

SCHEMBL21397973

c1ccc(-c2nc(-c3ccccc3)nc(-n3c4cnccc4c4ccc5c6ccccc6n(-c6ccccc6)c5c43)n2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.41
ATM Q13315 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
DYRK1A Q13627 1/20 0.38
CDK4 P11802 2/20 0.35
CDK6 Q00534 2/20 0.35
AOC3 Q16853 2/20 0.34
KCNH2 Q12809 1/20 0.34
REN P00797 1/20 0.34
KMT2A Q03164 3/20 0.34
MEN1 O00255 2/20 0.34
ALDH1A1 P00352 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C9 P11712 2/20 0.34
MAPT P10636 2/20 0.34
PDE5A O76074 2/20 0.34
HSP90AA1 P07900 1/20 0.34
GLA P06280 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21398001 1.00 KDM4E (0.41) KDM4EATML3MBTL1DYRK1ACDK4
SCHEMBL21397991 0.96 DYRK1A (0.40) DYRK1ACDK4CDK6AOC3KCNH2
SCHEMBL17349101 0.93 DYRK1A (0.39) KDM4EATML3MBTL1DYRK1ACDK4
SCHEMBL21397987 0.93 ATM (0.41) KDM4EATML3MBTL1RENKMT2A
SCHEMBL21397974 0.93 ATM (0.41) KDM4EATML3MBTL1RENKMT2A
SCHEMBL10029916 0.90 MEN1 (0.42) KDM4EATML3MBTL1KMT2AMEN1
SCHEMBL21397986 0.90 KDM4E (0.39) KDM4EATML3MBTL1DYRK1ACDK4
SCHEMBL126253 0.90 L3MBTL1 (0.50) KDM4EATML3MBTL1KMT2AMEN1
SCHEMBL30367723 0.90 L3MBTL1 (0.50) KDM4EATML3MBTL1KMT2AMEN1
SCHEMBL30021164 0.90 L3MBTL1 (0.50) KDM4EATML3MBTL1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019179497-A1 ORGANIC COMPOUND WITH PYRIDINE AS CORE AND USE THEREOF 江苏三月光电科技有限公司 2019-09-26 WO disclosed