SCHEMBL21407

SCHEMBL21407

Clc1cccc(COc2ccccc2)c1.OBO

nearest known ligand 0.66

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RXRA P19793 2/20 0.66
RXRB P28702 2/20 0.66
RXRG P48443 2/20 0.66
NR4A2 P43354 1/20 0.64
MAOB P27338 6/20 0.64
MAOA P21397 2/20 0.60
PKM P14618 1/20 0.58
GID4 Q8IVV7 1/20 0.55
ALOX5 P09917 1/20 0.55
NPC1 O15118 1/20 0.54
CYP1A2 P05177 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
RAB9A P51151 1/20 0.54
MRGPRX4 Q96LA9 1/20 0.54
ENPP2 Q13822 1/20 0.54
S1PR1 P21453 1/20 0.53
S1PR5 Q9H228 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11959143 0.93 MAOB (0.72) RXRARXRBRXRGNR4A2MAOB
Methyl Alcohol SCHEMBL9626623 0.92 RXRA (0.68) RXRARXRBRXRGNR4A2MAOB
Alcohol SCHEMBL9628500 0.89 RXRA (0.64) RXRARXRBRXRGNR4A2MAOB
Propanol SCHEMBL9627268 0.86 RXRA (0.61) RXRARXRBRXRGNR4A2MAOB
Isopropylamine SCHEMBL9628060 0.84 MAOB (0.65) RXRARXRBRXRGNR4A2MAOB
Ethylamine SCHEMBL9628064 0.84 MAOB (0.69) RXRARXRBRXRGNR4A2MAOB
SCHEMBL3624161 0.83 MAOB (0.73) RXRARXRBRXRGNR4A2MAOB
SCHEMBL3823697 0.82 RXRA (0.69) RXRARXRBRXRGNR4A2MAOB
Benzylphenylether SCHEMBL22314 0.82 LMNA (0.69) NR4A2MAOBMAOACYP1A2CYP2C19
SCHEMBL4698486 0.81 NR4A2 (0.66) RXRARXRBRXRGNR4A2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed