SCHEMBL21423976

SCHEMBL21423976

CC(=O)NCC(=O)CNC(=O)C(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
PTGS2 P35354 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
SOAT1 P35610 1/20 0.36
DPP4 P27487 1/20 0.36
PREP P48147 1/20 0.36
FAP Q12884 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MAPK1 P28482 1/20 0.36
HIF1A Q16665 1/20 0.36
ECE1 P42892 1/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C19 P33261 2/20 0.34
CYP2C9 P11712 1/20 0.34
KMT2A Q03164 1/20 0.34
ERCC1 P07992 1/20 0.34
ERCC4 Q92889 1/20 0.34
MME P08473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25514706 0.91 ALDH1A1 (0.44) ALDH1A1LMNAMAPTPTGS2TDP1
SCHEMBL5597209 0.83 KDM4E (0.48) ALDH1A1SOAT1DPP4PREPFAP
SCHEMBL25964962 0.79 ALDH1A1 (0.45) ALDH1A1LMNAMAPTPTGS2TDP1
SCHEMBL20991917 0.79 TDP1 (0.41) ALDH1A1LMNAMAPTPTGS2TDP1
SCHEMBL28497156 0.79 ALDH1A1 (0.40) ALDH1A1LMNAMAPTPTGS2TDP1
SCHEMBL10199485 0.78 ALDH1A1 (0.43) ALDH1A1LMNAMAPTPTGS2TDP1
SCHEMBL14015909 0.77 ALDH1A1 (0.39) ALDH1A1LMNAMAPTPTGS2TDP1
SCHEMBL10311745 0.76 MAPK1 (0.50) ALDH1A1MAPTKDM4EMAPK1HIF1A
SCHEMBL14069651 0.76 KDM4E (0.39) ALDH1A1LMNAMAPTPTGS2TDP1
SCHEMBL2608304 0.74 ALDH1A1 (0.40) ALDH1A1LMNAMAPTPTGS2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3778573-A1 COMPOUND WITH ANTICANCER ACTIVITY Kyowa Kirin Co., Ltd. (JP) 2021-02-17 EP disclosed
WO-2019189778-A1 COMPOUND WITH ANTICANCER ACTIVITY 協和発酵キリン株式会社 2019-10-03 WO disclosed