SCHEMBL21451816

SCHEMBL21451816

O=C(c1nc2c(s1)CN(CCOCCO)CC2)N1CCc2c(-c3cccc4c3CCN4C(=O)c3nc4c(s3)CN(CCSCCO)CC4)cccc21

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 16/20 0.39
CD274 Q9NZQ7 16/20 0.39
HDAC3 O15379 4/20 0.36
HDAC1 Q13547 4/20 0.36
HDAC6 Q9UBN7 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22966846 0.94 PDCD1 (0.43) PDCD1CD274HDAC3HDAC1HDAC6
SCHEMBL22966696 0.81 PDCD1 (0.42) PDCD1CD274HDAC3HDAC1HDAC6
SCHEMBL22966498 0.80 PDCD1 (0.41) PDCD1CD274HDAC3HDAC1HDAC6
SCHEMBL22966709 0.79 HDAC6 (0.42) PDCD1CD274HDAC3HDAC1HDAC6
SCHEMBL21451792 0.78 PDCD1 (0.45) PDCD1CD274HDAC3HDAC1HDAC6
SCHEMBL21451984 0.78 HDAC6 (0.44) PDCD1CD274HDAC3HDAC1HDAC6
SCHEMBL22966641 0.77 PDCD1 (0.44) PDCD1CD274HDAC3HDAC1HDAC6
SCHEMBL21451803 0.77 PDCD1 (0.42) PDCD1CD274
SCHEMBL22966819 0.76 PDCD1 (0.42) PDCD1CD274
SCHEMBL21452331 0.76 ROCK2 (0.46) PDCD1CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019192506-A1 IMMUNOMODULATORS, COMPOSITIONS AND METHODS THEREOF BETTA PHARMACEUTICALS CO., LTD (CN) 2019-10-10 WO disclosed