SCHEMBL21452006

SCHEMBL21452006

N#Cc1cc(C2(N)CCCC(O)C2=O)ccc1C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AR P10275 15/20 0.39
TRPA1 O75762 1/20 0.38
SLC22A12 Q96S37 1/20 0.35
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
TACR1 P25103 1/20 0.34
CYP2C19 P33261 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL21436242 0.96 AR (0.36) ARTRPA1SLC22A12CYP2D6CYP2C9
Oxalic Acid SCHEMBL30829178 0.96 AR (0.36) ARTRPA1SLC22A12CYP2D6CYP2C9
SCHEMBL21436244 0.84 AR (0.34) ARTRPA1SLC22A12CYP2D6CYP2C9
SCHEMBL30829164 0.83 PDE2A (0.40)
SCHEMBL21436149 0.83 PDE2A (0.40)
Hydrochloric Acid SCHEMBL28903253 0.82 PDE2A (0.39)
SCHEMBL21452004 0.78 SLC22A12 (0.38) ARTRPA1SLC22A12CYP2D6CYP2C9
SCHEMBL23002147 0.77 MAOA (0.41)
SCHEMBL21436185 0.77 MAOA (0.41)
SCHEMBL21436156 0.77 MAOA (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210171487-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF SHANGHAI JIANHE PHARMACEUTICAL & TECHNOLOGY CO. LTD. (CN) 2021-06-10 US disclosed
EP-3778579-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Jianhe Pharmaceutical & Technology Co. Ltd. (CN) 2021-02-17 EP disclosed
WO-2019192602-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海键合医药科技有限公司 2019-10-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210171487-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF CYP4F11, PAH, COMT AR 1775/4885TRPA1 278/4885SLC22A12 692/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.