SCHEMBL21452373

SCHEMBL21452373

Cc1cccc(C2(NC(=O)OC(C)(C)C)CC(C)CCC2=O)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.38
GPR119 Q8TDV5 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
CCKBR P32239 1/20 0.35
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
BRD4 O60885 1/20 0.34
CREBBP Q92793 1/20 0.34
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
HDAC4 P56524 1/20 0.34
EPHX2 P34913 1/20 0.34
EGFR P00533 1/20 0.34
PRKACA P17612 1/20 0.34
FRK P42685 1/20 0.34
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
NEK4 P51957 1/20 0.34
PRKCD Q05655 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21452404 0.88 MEN1 (0.42) MEN1KMT2ACCKBREPHX2ALDH1A1
SCHEMBL21452126 0.82 RORC (0.41) CCR2
SCHEMBL21452370 0.82 HDAC4 (0.47) GPR119MEN1KMT2AOPRM1HDAC4
SCHEMBL23003282 0.82 RORC (0.41) CCR2
SCHEMBL23001555 0.81 PDE2A (0.39) HDAC4MAPTALDH1A1TDP1
SCHEMBL21452417 0.81 PDE2A (0.39) HDAC4MAPTALDH1A1TDP1
SCHEMBL21451897 0.79 HDAC4 (0.39) GPR119MEN1KMT2ACCKBRHCRTR1
SCHEMBL21452464 0.78 DPP8 (0.35) MEN1KMT2ABRD4CREBBPDDB1
SCHEMBL21452507 0.74 SCN9A (0.35) BRD4CREBBPEPHX2DDB1CRBN
SCHEMBL21452508 0.74 SCN9A (0.35) BRD4CREBBPEPHX2DDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019192602-A1 AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海键合医药科技有限公司 2019-10-10 WO disclosed